Synthesis and evaluation
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The outcomes are to be compared with typical drugs given that compounds are examined against gram-positive and gram-negative strains of bacteria and fungus. Against bacterial strains, products with nitro, methyl, and bromo substituents in the p-position of the benzene ring, as well as products with the nitro group at the m-position, showed very excellent activities against bacterial strains, while compounds with chloro substituent at p-position and m-position demonstrated good activity against the fungal strains Aspergillus niger and Fusarium javanicum.
8p dianmotminh02 03-05-2024 5 1 Download
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The present study focuses on the preparation of silver/copper bimetallic hybrid nanoparticles by green method from precursor solutions of silver nitrate & copper nitrate and the locally available citrus fruit (lemon) peel extract which behaves as the stabilizing and reducing agent. Initially, the formation of hybrid nanoparticles was noticed in the reaction mixture by colour change.
7p dianmotminh02 03-05-2024 4 1 Download
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This article, we present a thorough and straightforward hydrothermal method towards the production of reduced graphene oxide templated MIL-53(Fe) hybrids RGO@MIL-53(Fe). The structural characteristics of created hybrids were identified by using BET, FESEM, powder X-ray diffraction, and FTIR techniques. Methylene blue (MB) dye (a model water pollutant) was used to evaluate H2O2-assisted photo-catalytic efficiency of RGO@MIL-53(Fe).
9p dianmotminh02 03-05-2024 2 1 Download
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. In vitro biological evaluation revealed the most active compound 4d with an inhibitory concentration of 42.87 μM against K562 and 47.42 μM on A549 cells. The anticancer activity of this naphthylidene isoxazolidinedione derivative was evident by cell cycle and apoptosis assays, which showed arrest of the G2/M phase (65.6%) of the K562 cells and induction of apoptosis with 21.47% apoptotic cells as compared to 0.2% of untreated cells, respectively.
10p dianmotminh02 03-05-2024 5 3 Download
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natural fiber for the construction of hybrid bio-composites. In the current research project, a thorough analysis of the use of soy-PF resin for the creation of composites reinforced with jute was conducted. A novel and practical cutlery material was created after the mechanical properties were evaluated and optimized. In order to study the value addition of these newly proposed biocomposite materials as an ecological alternative in terms of natural resources versus synthetic resources, variables such as hardness, cytotoxicity, and degrading qualities of composites were also explored.
9p dianmotminh02 03-05-2024 5 2 Download
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The aim of our in vitro study was to assess the potential effect of BPF on H295R cells mitochondrial activity, metabolic activity, membrane integrity, lysosomal function, and testosterone synthesis. Adrenocortical carcinoma cells were cultivated during 24 h in the presence of BPF (0.1, 0.5, 1, 10, 25, 50, 75, 100, 300, 500 μM). Exposure doses of BPF caused a significant decrease of mitochondrial activity starting from 1 μM, we observed a slight increase in mitochondrial activity at the lowest concentration (0.1 μM).
4p mudbound 10-12-2021 11 1 Download
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The purpose of this thesis is to study and synthesize BiMO materials (M = V,Ti,Sn) by microwaveassisted chemical method, hydrothermal method, sol-gel method and evaluate their physical properties. The synthesized materials (Bi2Sn2O7 and Bi2Ti2O7) were investigated the photocatalytic activity in the decomposition of RhotaminB (RhB) under visible light.
28p thebadguys 08-06-2021 22 3 Download
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Objectives of the dissertation: Research and synthesize and determine the hybrid compound structure containing Quinazoline frame. Research on carcinogenic activity and inhibition of acetylcholinesterase enzyme of synthetic compounds..
26p extraenglish 24-05-2021 21 3 Download
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Aim of the thesis: Synthesis of several derivatives and tubulysin analogues with the replacement of the amino acid methylpipecolic (Mep) at the N-terminal, replacing N,O-acetyl group by methyl group, and researching the role of tubuphenylalanine (Tup) group at the C-terminal.
26p extraenglish 24-05-2021 14 3 Download
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Synthesis and structural determination of some 4-aminoquinazoline derivatives containing prop-2-yn-1-yloxy substituents at C-6 position; research and synthesize and determine the hybrid compound structure containing Quinazoline frame; research on carcinogenic activity and inhibition of acetylcholinesterase enzyme of synthetic compounds; studying protein docking and predicting the pharmacokinetic properties of some compounds that inhibit the enzyme acetylcholinesterase.
26p capheviahe27 23-02-2021 36 4 Download
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Synthesis of several derivatives and tubulysin analogues with the replacement of the amino acid methylpipecolic (Mep) at the N-terminal, replacing N,O-acetyl group by methyl group, and researching the role of tubuphenylalanine (Tup) group at the C-terminal .
26p capheviahe27 23-02-2021 17 5 Download
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The thesis focused on the synthesis of Mn, Ce, C doped ZnO nanoparticles materials and doped ZnO with multi-layered carbon nanotube nanocomposite materials and assessed their photo-oxidative potentiality through photocatalytic reactions of methylene blue (MB) decomposition in aqueous solution under visible light.
30p capheviahe27 23-02-2021 19 4 Download
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Successfully synthesized nano – mixed oxide by different gelling agents; compared, selected the appropriate gelling agent; researched to evaluate the catalytic activity of mixed oxide nanoparticles formed with pollutants methyl orange (MO), methylene blue (MB). Successful dispersed mixed oxide nanoparticles on rGO; investigated catalytic activity of material systems on parathion, fenitrothion.
28p capheviahe26 25-01-2021 30 5 Download
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Usnic acid isolated from lichen was a potential bioactivity compound. It has a broad spectrum bioactivity, including antiviral, anti-inflammatory, anticancer… However, low solubility in water limited its application. Many researchs have done to overcome the restriction. Recent results showed that usnic acid derivatives bearing triazole, enamine, pyrazole and benzylidene groups had strong antiviral and anticancer activities. Thus, investigation of usnic acid derivatives synthesis was an attractive aspect due to the diversity of bioactivities of usnic acid derivatives.
8p larachdumlanat127 02-01-2021 5 1 Download
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A series of semicarbazones, thiosemicarbazones, 1,3,4-oxadiazoles/thiadiazoles bearing pyrazole scaffold were designed and synthesized. All the synthesized new compounds were characterized by 1H NMR, 13C NMR, MS and elemental analysis.
14p tocectocec 26-05-2020 28 2 Download
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The presence of heterocyclic moiety in diverse compounds, strongly indicative of the desired effect on physiological activity, and it reflects on efforts to find useful synthetic drugs.
12p tocectocec 25-05-2020 13 0 Download
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Antimicrobial resistance is an emerging challenge for health personnel and researchers. In such scenario, alternative strategies targeting novel ways to kill or inhibit growth of microbes are need of the hour. Antimicrobial peptide can be a promising candidate to deal with this crisis. Extracellular matrix protein vitronectin (Vn) is recently being established as a bactericidal agent against certain microbes. Caprine Vn has got few structural alterations as compare to human Vn.
7p nguaconbaynhay5 16-05-2020 13 0 Download
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The objectives of the thesis: The thesis focused on the synthesis of Mn, Ce, C doped ZnO nanoparticles materials and doped ZnO with multi-layered carbon nanotube nanocomposite materials and assessed their photo-oxidative potentiality through photocatalytic reactions of methylene blue (MB) decomposition in aqueous solution under visible light.
30p phongtitriet000 08-08-2019 42 4 Download
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The objectives of the thesis: Synthesis of new vinca alkaloid derivatives containing different substituents on C-3' and N-6' positions in ring D of the velbanamine subunit, concurrently evaluating the biological activity of the derivatives synthesized.
27p xacxuoc4321 09-07-2019 22 5 Download
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Main contents of thesis: Introdution of fuel cell and studies on Pt catalysts and Pt alloy catalysts in PEMFC. Research on synthesis of catalytic materials Pt/C 20% wt. by electroless deposition method and evaluating to influence of experimental parameters such as pH, temperature... in the synthesis process on the properties of catalyst Pt / C 20%wt.
22p xacxuoc4321 09-07-2019 48 4 Download